2021-2022 Graduate Catalog

CH 526 Medicinal Chemistry & Pharmacology

A basic medicinal chemistry/pharmacology course in which the principles of drug discovery, computer aided drug design, pharmacokinetics and protein targets are studied.  Such topics as the background of drug discovery, protein structure, enzymes, receptors, pharmacokinetics, metabolism, binding, structure, diversity, lead discovery, and lead optimization.  Different methods to design drugs are explored such as rational drug design, fragment based, and in silico virtual molecular docking.  Virtual labs employing different software are used to exemplify the different concepts covered.

Credits

3